Cytotoxicity of isoflavones from Millettia dura

Loading...
Thumbnail Image

Date

2019

Authors

Buyinza, Daniel
Yang, Li Jun
Derese, Solomon
Ndakala, Albert
Coghi, Paolo
Heydenreich, Matthias
Wong, Vincent Kam Wai
Möller, Heiko M.
Yenesew, Abiy

Journal Title

Journal ISSN

Volume Title

Publisher

Taylor & Francis

Abstract

The first phytochemical investigation of the flowers of Millettia dura resulted in the isolation of seven isoflavones, a flavonol and a chalcone. Eleven isoflavones and a flavonol isolated from various plant parts from this plant were tested for cytotoxicity against a panel of cell lines, and six of these showed good activity with IC50 values of 6-14 lM. Durmillone was the most active with IC50 values of 6.6 lM against A549 adenocarcinomic human alveolar basal epithelial cancer cell line with low cytotoxicity against the non-cancerous cell lines BEAS-2B (IC50 ¼ 58.4 lM), LO2 hepatocytes (IC50 78.7 lM) and CCD19Lu fibroblasts (IC50 >100 lM).

Description

Keywords

Millettia dura, Leguminosae, isoflavone, cytotoxicity

Citation

Daniel Buyinza, Li Jun Yang, Solomon Derese, Albert Ndakala, Paolo Coghi, Matthias Heydenreich, Vincent Kam Wai Wong, Heiko M. Möller & Abiy Yenesew (2019): Cytotoxicity of isoflavones from Millettia dura, Natural Product Research, DOI: 10.1080/14786419.2019.1660335